neurotensin receptor - Robuta Search

https://pubmed.ncbi.nlm.nih.gov/19195889/

The identification of nonpeptide neurotensin receptor partial agonists from the potent antagonist...

In a search for nonpeptide agonists for the neurotensin receptor (NTR1), we replaced the adamantyl amino acid moiety found in the antagonist SR48692 (1a) with...

neurotensin receptor partial agonists identification nonpeptide

https://www.ncbi.nlm.nih.gov/Structure/pdb/6PWC

6PWC: A complex structure of arrestin-2 bound to neurotensin receptor 1

Beta-arrestin-1Fab30 heavy chainFab30 light chainNeurotensin peptideNeurotensin receptor type 1

complex structure arrestin bound neurotensin

https://www.preprints.org/manuscript/202306.2214

Mechanistic Elucidation of Activation/Deactivation Signal Transduction within Neurotensin Receptor...

Small molecule modulators of neurotensin receptor 1 (NTSR1), a class A G protein-coupled receptor (GPCR), has been emerging as promising therapeutics for...

signal transduction neurotensin receptor mechanistic elucidation activation

https://www.rcsb.org/structure/6UP7

RCSB PDB - 6UP7: neurotensin receptor and arrestin2 complex

neurotensin receptor and arrestin2 complex

rcsb pdb neurotensin receptor complex