https://www.cas.org/resources/webinar/webinar-bond-worth-forming-rise-targeted-covalent-inhibitors
Webinar: A Bond Worth Forming: The Rise of Targeted Covalent Inhibitors | CAS
Join our expert panel to explore targeted covalent inhibitors, their role in addressing challenging targets, and insights into the inhibitor landscape.
targeted covalent inhibitorsthe rise
https://elifesciences.org/reviewed-preprints/101401
Targeted anticancer pre-vinylsulfone covalent inhibitors of carbonic anhydrase IX
covalent inhibitorscarbonic anhydrasetargetedanticancerpre
https://elifesciences.org/articles/101401
Targeted anticancer pre-vinylsulfone covalent inhibitors of carbonic anhydrase IX | eLife
A series of compounds were synthesized and demonstrated to form a specific covalent bond with His64 of CAIX, an anticancer target, a strategy applicable to any...
carbonic anhydrase ixcovalent inhibitorstargetedanticancerpre
https://pmc.ncbi.nlm.nih.gov/articles/PMC9827112/
Creating MHC-Restricted Neoantigens with Covalent Inhibitors That Can Be Targeted by Immune Therapy...
Cancer-specific neoantigens created in the form of a covalent drug conjugated to a fragment of an intracellular oncoprotein selectively mark drug-resistant...
https://elifesciences.org/reviewed-preprints/101401v1/reviews
Targeted anticancer pre-vinylsulfone covalent inhibitors of carbonic anhydrase IX
covalent inhibitorscarbonic anhydrasetargetedanticancerpre