Robuta

https://www.ncbi.nlm.nih.gov/Structure/pdb/5D3S 5D3S: First bromodomain of BRD4 bound to inhibitor XD44 Bromodomain-containing protein 4(R,R)-2,3-BUTANEDIOL4-acetyl-3-ethyl-N-[4-fluoro-3-(morpholin-4-ylsulfonyl)phenyl]-5-methyl-1H-pyrrole-2-carboxamideDIMETHYL... firstbromodomainboundinhibitor