https://www.techtransfer.nih.gov/patent/e-290-1997-0-it-11
G-PROTEIN-COUPLED RECEPTOR ANTAGONISTS | Technology Transfer
g proteinreceptor antagonistscoupledtechnologytransfer
https://experts.umn.edu/en/publications/mineralocorticoid-receptor-antagonists-as-diuretics-can-congestiv/
Mineralocorticoid receptor antagonists as diuretics: Can congestive heart failure learn from liver...
congestive heart failuremineralocorticoid receptor
https://www.techtransfer.nih.gov/patent/e-285-2008-0-pct-02
Truncated (N)-Methanocarba Adenosine Derivatives As A3 Receptor Antagonists | Technology Transfer
receptor antagonistsadenosinederivatives
https://gpe.wikipedia.org/wiki/Category:Glycine_receptor_antagonists
Category:Glycine receptor antagonists - Wikipedia
receptor antagonistscategoryglycinewikipedia
https://www.techtransfer.nih.gov/patent/e-028-2018-1-hk-08
HETEROCYCLIC P2Y14 RECEPTOR ANTAGONISTS | Technology Transfer
receptor antagonistsheterocyclictechnologytransfer
https://adisinsight.springer.com/drugs/800086816?error=cookies_not_supported&code=f5485e31-97c3-4d19-a6a7-357f723e074c
Calcitonin gene related peptide receptor antagonists - Pfizer - AdisInsight
Pfizer is developing a calcitonin gene related peptide (CGRP) receptor antagonists for the treatment of undisclosed indication. Clinical development is underway
receptor antagonistscalcitoningenerelatedpeptide
https://www.techtransfer.nih.gov/patent/e-096-1998-0-ca-03
A3 Adenosine Receptor Antagonists | Technology Transfer
adenosine receptorantagoniststechnologytransfer
https://research.birmingham.ac.uk/en/publications/qualitative-and-quantitative-simulation-of-androgen-receptor-anta/fingerprints/
Qualitative and quantitative simulation of androgen receptor antagonists: A case study of...
androgen receptorqualitativequantitativesimulation
https://publications-cnrc.canada.ca/fra/voir/objet/?id=cb3fa8d6-5087-4aaf-a459-14da092fd504
Glutamate receptor antagonists for the treatment of cerebral ischemia - Archives des publications...
Glutamate receptor antagonists for the treatment of cerebral ischemia
receptor antagonistsfor the
https://pubchem.ncbi.nlm.nih.gov/patent/EP-0479481-A3
Fibrinogen receptor antagonists - Patent EP-0479481-A3 - PubChem
EP-0479481-A3 chemical patent summary.
receptor antagonistsfibrinogenpatentpubchem
https://adisinsight.springer.com/drugsafety/800007631?error=cookies_not_supported&code=f3455bba-8a92-4a33-b986-45317a2b7ed2
Comparable safety profiles of the H2-receptor antagonists - AdisInsight
Despite the excellent safety record of the H2-receptor antagonists, cimetidine, ranitidine, famotidine and nizatidine, there remains a degree of confusion
of thereceptor antagonistscomparablesafetyprofiles
https://www.techtransfer.nih.gov/patent/e-213-2015-0-us-05
TRIAZOLE DERIVATIVES AS P2Y14 RECEPTOR ANTAGONISTS | Technology Transfer
triazole derivativesreceptor antagoniststechnologytransfer
https://experts.colorado.edu/display/meshid_D27.505.519.364
Endothelin Receptor Antagonists | CU Experts | CU Boulder
endothelin receptorantagonistscuexpertsboulder
https://www.techtransfer.nih.gov/patent/e-162-2023-0-pc-01
5-HT2B SEROTONIN RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITIONS THEREOF, AND METHODS OF USE...
receptor antagonists
https://adisinsight.springer.com/drugs/800046251?error=cookies_not_supported&code=f8a517d3-0b19-46c6-bf4e-e31cbfe91a41
Research programme: mitochondrial angiotensin receptor antagonists - Gemstone Biotherapeutics -...
Gemstone Biotherapeutics LLC was developing mitochondrial angiotensin receptor antagonists, utilising discoveries and technologies pioneered by researchers at
research programmeangiotensin receptormitochondrialantagonistsgemstone
https://www.wikidata.org/wiki/Q40661137
Antigen analogs/MHC complexes as specific T cell receptor antagonists - Wikidata
scientific article published on January 1994
mhc complexest cellreceptor antagonistsantigenanalogs
https://adisinsight.springer.com/drugsafety/803930138?error=cookies_not_supported&code=20e212ed-875b-4c8a-a261-8eeefb4245c5
Programmed cell death 1 receptor antagonists - AdisInsight
A patient receiving PD-1 inhibitor treatment experienced an atypical Herpes simplex-2 infection.
cell deathreceptor antagonistsprogrammedadisinsight
https://www.techtransfer.nih.gov/patent/e-285-2008-0-de-08
A3 Adenosine Receptor Antagonists and Partial Agonists | Technology Transfer
adenosine receptorantagonistspartialtechnologytransfer
https://adisinsight.springer.com/drugsafety/803929520?error=cookies_not_supported&code=a2538174-c6a0-4393-894c-d0498f816163
Programmed cell death 1 receptor antagonists - AdisInsight
Three patients with recurrent or metastatic maxillary sinus squamous cell carcinoma [ages and sexes not stated] were included among 15 individuals treated at
cell deathreceptor antagonistsprogrammedadisinsight
https://www.sciencedaily.com/releases/2021/11/211108094235.htm
Healing skin ischemia-reperfusion injuries with interleukin-36 receptor antagonists | ScienceDaily
Skin wounds from ischemia-reperfusion injuries -- tissue damage caused by blood returning to tissues after a period of oxygen deprivation -- may not heal...
receptor antagonistshealingskinischemiareperfusion
https://pubmed.ncbi.nlm.nih.gov/28864614/
Somatostatin Receptor Antagonists for Imaging and Therapy
Somatostatin receptor (sstr) scintigraphy for imaging and sstr analogs for treatment have been used for more than 20 y. An important improvement in recent...
somatostatin receptorantagonistsimagingtherapy
https://www.techtransfer.nih.gov/patent/e-213-2001-0-us-01
Anticancer Effects of a Novel Vitamin D Receptor Antagonists | Technology Transfer
vitamin d receptoranticancereffectsnovel
https://adisinsight.springer.com/drugsafety/803928660?error=cookies_not_supported&code=10916989-d921-423b-86d2-9c05024aeabe
Programmed cell death 1 receptor antagonists - AdisInsight
Five patients [ages and sexes not stated] treated with anti-programmed death-1 (PD-1) immune checkpoint inhibition [route, dosage and duration not stated]
cell deathreceptor antagonistsprogrammedadisinsight
https://adisinsight.springer.com/drugsafety/803928181?error=cookies_not_supported&code=5772ef7a-ef63-41bf-afa9-b94bf346678c
Immune checkpoint protein inhibitors/Programmed cell death 1 receptor antagonists - AdisInsight
Fifty-nine adult patients [exact ages and sexes not stated] with cancer who received immune checkpoint inhibitors [dose, route and treatment duration not
immune checkpointcell deathreceptor antagonistsproteininhibitors
https://pmc.ncbi.nlm.nih.gov/articles/PMC17685/
SST3-selective potent peptidic somatostatin receptor antagonists - PMC
A family of octapeptide derivatives of somatostatin cyclized via a disulfide bridge (des-AA1,2,4,5,12,13[d-2Nal8]-somatostatin-14, ODN-8) was identified that...
somatostatin receptorselectivepotentantagonistspmc
https://pubmed.ncbi.nlm.nih.gov/10416935/
Effects of muscarinic cholinergic receptor antagonists on postnatal eye growth of rhesus monkeys
The drug treatment results implicate muscarinic receptors in postnatal eye growth regulation. Because of interanimal differences our data do not indicate...
receptor antagonists
https://www.techtransfer.nih.gov/patent/e-028-2018-1-ca-03
HETEROCYCLIC P2Y14 RECEPTOR ANTAGONISTS | Technology Transfer
receptor antagonistsheterocyclictechnologytransfer
https://www.techtransfer.nih.gov/patent/e-051-2021-0-us-02
HETEROCYCLIC P2Y14 RECEPTOR ANTAGONISTS | Technology Transfer
receptor antagonistsheterocyclictechnologytransfer
https://experts.colorado.edu/display/meshid_D27.505.519.625.240.300.500
Molecular Mechanisms of Pharmacological Action - GABA-A Receptor Antagonists | CU Experts | CU...
receptor antagonistsmolecularmechanismspharmacologicalaction
https://about.uq.edu.au/experts/project/45180
Characterisation of the effect of C5a receptor antagonists against the C5a-like receptor 2 (C5L2) |...
of thereceptor antagonistscharacterisationeffect
https://grillbert.substack.com/p/nmda-receptor-antagonists-a-bit-more/comments
Comments - NMDA Receptor Antagonists: Slightly More than you Wanted to Know
Insights from Memantine and Ketamine's divergent effects on the Brain
nmda receptor antagonistsmore thancommentsslightly
https://pubchem.ncbi.nlm.nih.gov/patent/EP-1146872-B1
Use of angiotensin ii receptor antagonists for treating acute myocardial infarction - Patent...
EP-1146872-B1 chemical patent summary.
acute myocardial infarctionangiotensin iireceptor antagonists
https://www.techtransfer.nih.gov/patent/e-285-2008-0-us-07
A3 Adenosine Receptor Antagonists And Partial Agonists | Technology Transfer
adenosine receptorantagonistspartialtechnologytransfer
https://www.cochrane.org/zh-hant/evidence/CD005449_adenosine-diphosphate-adp-receptor-antagonists-prevention-cardiovascular-disease-patients-type-2
Adenosine-diphosphate (ADP) receptor antagonists for the prevention of cardiovascular disease in...
receptor antagonistsfor the
https://hsrc.himmelfarb.gwu.edu/gwhpubs/2138/
"Nonsteroidal mineralocorticoid receptor antagonists and cardiorenal ou" by Kevin Bryan Lo, Janani...
The burden of adverse cardiorenal outcomes among patients with the trifecta of diabetes, heart failure (HF), and chronic kidney disease (CKD) remains high....
mineralocorticoid receptor
https://cebs-ext.niehs.nih.gov/datasets/search/androgen_antagonists?casrn=30560-19-1
Evaluation of Androgen Receptor Antagonists | DTT Data Collections Guided Search
androgen receptordata collectionsevaluationantagonistsdtt
https://nrc-publications.canada.ca/eng/view/object/?id=99b40bc6-8fda-4466-b27f-73323f96365a
Excitotoxicity and glutamate receptor antagonists in Neuroprotection - NRC Publications Archive -...
Excitotoxicity and glutamate receptor antagonists in Neuroprotection
receptor antagonistsexcitotoxicityglutamateneuroprotectionnrc
https://www.techtransfer.nih.gov/patent/e-235-2008-0-us-01
P2Y1 RECEPTOR ANTAGONISTS | Technology Transfer
receptor antagoniststechnologytransfer
https://adisinsight.springer.com/drugsafety/803927857?error=cookies_not_supported&code=e6eb660f-8439-4d74-98e7-67af8387a3e2
Disitamab vedotin/Programmed cell death 1 receptor antagonists - AdisInsight
Twenty-nine patients with metastatic urothelial carcinoma, with a reported median age of 67 years and predominantly male (69%), received disitamab vedotin
cell deathreceptor antagonistsprogrammedadisinsight
https://vivo.colorado.edu/display/pubid_52302
THE BENZODIAZEPINE RECEPTOR ANTAGONISTS FLUMAZENIL AND CGS8216 BLOCK THE ENHANCEMENT OF FEAR...
receptor antagonistsbenzodiazepineflumazenil
https://www.aafp.org/pubs/afp/issues/2003/0715/p354a.html
Leukotriene Receptor Antagonists vs. Steroids | AAFP
leukotriene receptorantagonistsvssteroidsaafp
https://www.techtransfer.nih.gov/patent/e-310-2005-0-us-01
Prodrug Delivery Of A3 Adenosine Receptor Antagonists For Glaucoma Therapy | Technology Transfer
adenosine receptor
https://www.techtransfer.nih.gov/patent/e-213-2015-0-gb-08
TRIAZOLE DERIVATIVES AS P2Y14 RECEPTOR ANTAGONISTS | Technology Transfer
triazole derivativesreceptor antagoniststechnologytransfer
https://experts.arizona.edu/en/publications/pharmacology-of-modality-specific-transient-receptor-potential-va/
Pharmacology of modality-specific transient receptor potential vanilloid-1 antagonists that do not...
https://www.techtransfer.nih.gov/patent/e-226-1992-0-be-05
Methods for the Improvement of Cognition with Functional Antagonists of the Glycine NMDA Receptor...
for the
https://experts.arizona.edu/en/publications/transient-receptor-potential-vanilloid-1-antagonists-prevent-anes/
Transient Receptor Potential Vanilloid 1 Antagonists Prevent Anesthesia-induced Hypothermia and...
transientreceptorpotential
https://lnu.diva-portal.org/smash/record.jsf?pid=diva2:308572
Potency mismatch for behavioral and biochemical effects by dopamine receptor antagonists:...
dopamine receptorpotencymismatchbehavioral
https://vivo.colorado.edu/display/meshid_D27.505.519.625.850.850.200
Molecular Mechanisms of Pharmacological Action - Serotonin 5-HT2 Receptor Antagonists | CU Experts...
https://profiles.wustl.edu/en/publications/design-and-synthesis-of-amidino-tyrosine-derivatives-as-non-pepti/
Design and synthesis of amidino-tyrosine derivatives as non-peptide fibrinogen receptor antagonists...
https://www.techtransfer.nih.gov/patent/e-191-1993-3-de-05
A3 ADENOSINE RECEPTOR AGONISTS AND ANTAGONISTS | Technology Transfer
adenosine receptor agonistsantagoniststechnologytransfer
https://pure.psu.edu/en/publications/potential-anxiogenic-effects-of-cannabinoid-cb1-receptor-antagoni/
Potential anxiogenic effects of cannabinoid CB1 receptor antagonists/inverse agonists in rats:...
https://www.techtransfer.nih.gov/patent/e-253-1999-1-ep-08
USE OF A3 ADENOSINE RECEPTOR ANTAGONISTS IN THE MANUFACTURE OF A MEDICAMENT FOR REDUCING...
https://www.techtransfer.nih.gov/patent/e-226-1992-0-ie-12
Methods for the Improvement of Cognition with Functional Antagonists of the Glycine NMDA Receptor...
for the
https://pmc.ncbi.nlm.nih.gov/articles/PMC10325868/
Daridorexant, a Recently Approved Dual Orexin Receptor Antagonists (DORA) in Treatment of Insomnia...
Insomnia is one of the major challenges in medical science nowadays as it leads to great socio-economic burden by impairing daytime function as well as the...
https://research.monash.edu/en/publications/intravitreal-administration-of-endothelin-type-a-receptor-or-endo/
Intravitreal administration of endothelin type A receptor or endothelin type B receptor antagonists...
type aadministrationreceptorbantagonists
https://pubchem.ncbi.nlm.nih.gov/bioassay/2357
AID 2357 - SAR Analysis of Antagonists of the DOR Receptor using an Image-Based Assay - PubChem
BioAssay record AID 2357 submitted by Sanford-Burnham Center for Chemical Genomics: SAR Analysis of Antagonists of the DOR Receptor using an Image-Based Assay.
https://pubmed.ncbi.nlm.nih.gov/30404914/
Structure-guided development of selective M3 muscarinic acetylcholine receptor antagonists
Drugs that treat chronic obstructive pulmonary disease by antagonizing the M3 muscarinic acetylcholine receptor (M3R) have had a significant effect on health,...
structureguideddevelopmentselectiveacetylcholine
https://www.techtransfer.nih.gov/patent/e-067-2010-0-ep-06
Inverse Agonists And Neutral Antagonists For the TSH Receptor | Technology Transfer
for thetsh receptorinverseagonistsneutral
https://www.techtransfer.nih.gov/patent/e-191-1993-3-it-09
A3 ADENOSINE RECEPTOR AGONISTS AND ANTAGONISTS | Technology Transfer
adenosine receptor agonistsantagoniststechnologytransfer
https://pmc.ncbi.nlm.nih.gov/articles/PMC3926345/
Long-acting muscarinic receptor antagonists for the treatment of chronic airway diseases - PMC
Acetylcholine (neuronal and non-neuronal origin) regulates bronchoconstriction, and mucus secretion. It has an inflammatory effect by inducing attraction,...
https://www.techtransfer.nih.gov/patent/e-121-1993-0-pct-02
8-SUBSTITUTED 1,3,7-TRIALKYL-XANTHINE DERIVATIVES AS A2-SELECTIVE ADENOSINE RECEPTOR ANTAGONISTS |...
https://oru.diva-portal.org/smash/record.jsf?faces-redirect=true&language=sv&searchType=SIMPLE&query=&af=%5B%5D&aq=%5B%5B%5D%5D&aq2=%5B%5B%5D%5D&aqe=%5B%5D&pid=diva2%3A1553229&noOfRows=50&sortOrder=author_sort_asc&sortOrder2=title_sort_asc&onlyFullText=false&sf=all
In silico and in vitro assessment of androgen receptor antagonists
in silicoandrogen receptorvitroassessmentantagonists
https://pubchem.ncbi.nlm.nih.gov/bioassay/1224840
AID 1224840 - qHTS assay to identify small molecule antagonists of the estrogen related receptor...
BioAssay record AID 1224840 submitted by Tox21: qHTS assay to identify small molecule antagonists of the estrogen related receptor signaling pathway with the...
https://pubchem.ncbi.nlm.nih.gov/patent/US-2008287398-A1
Cold menthol receptor-1 antagonists - Patent US-2008287398-A1 - PubChem
US-2008287398-A1 chemical patent summary.
patent uscoldmentholreceptorantagonists
https://pubchem.ncbi.nlm.nih.gov/bioassay/602448
AID 602448 - qHTS for antagonists of the Thyroid Stimulation Hormone Receptor: Hit Validation with...
BioAssay record AID 602448 submitted by National Center for Advancing Translational Sciences (NCATS): qHTS for antagonists of the Thyroid Stimulation Hormone...
https://www.techtransfer.nih.gov/patent/e-067-2010-0-au-03
Inverse Agonists And Neutral Antagonists For the TSH Receptor | Technology Transfer
for thetsh receptorinverseagonistsneutral
https://www.techtransfer.nih.gov/news/licensing-collaboration-opportunity-for-next-gen-5-ht-2b-serotonin-receptor-antagonists-for
Licensing/Collaboration Opportunity for Next-Gen 5-HT-2B Serotonin-Receptor Antagonists for...
collaboration opportunitynext gen
https://pubchem.ncbi.nlm.nih.gov/bioassay/1259247
AID 1259247 - qHTS assay to identify small molecule antagonists of the androgen receptor (AR)...
BioAssay record AID 1259247 submitted by Tox21: qHTS assay to identify small molecule antagonists of the androgen receptor (AR) signaling pathway using the MDA...
https://pubchem.ncbi.nlm.nih.gov/bioassay/2836
AID 2836 - SAR analysis of antagonists of the Cannabinoid Receptor 2 using an Image-Based Assay -...
BioAssay record AID 2836 submitted by Sanford-Burnham Center for Chemical Genomics: SAR analysis of antagonists of the Cannabinoid Receptor 2 using an...
https://www.techtransfer.nih.gov/patent/e-067-2010-0-in-07
Inverse Agonists And Neutral Antagonists For the TSH Receptor | Technology Transfer
for thetsh receptorinverseagonistsneutral
https://pubmed.ncbi.nlm.nih.gov/17479101/?dopt=Abstract
Therapeutic targeting of innate immunity with Toll-like receptor agonists and antagonists
The identification of the antigen recognition receptors for innate immunity, most notably the Toll-like receptors, has sparked great interest in therapeutic...
innate immunity
https://www.techtransfer.nih.gov/patent/e-053-2016-0-us-01
Dopamine D3 Receptor Selective Antagonists/Partial Agonists; Method of Making; and Use Thereof |...
https://pubmed.ncbi.nlm.nih.gov/33682527/
Pilot study of tolerability and safety of opioid receptor antagonists as novel therapies for...
ClinicalTrials.gov identifier: NCT03278886.
https://www.ncbi.nlm.nih.gov/Structure/pdb/5FQS
5FQS: Selective estrogen receptor downregulator antagonists: Tetrahydroisoquinoline phenols 3
ESTROGEN RECEPTOR(E)-3-[4-(6-HYDROXY-2-ISOBUTYL-1-METHYL-3,4-DIHYDROISOQUINOLIN-1-YL)PHENYL]PROP-2-ENOIC ACID
estrogen receptorselectiveantagonistsphenols
https://www.techtransfer.nih.gov/patent/e-323-2002-0-gb-05
USE OF A3 ADENOSINE RECEPTOR ANTAGONISTS IN THE MANUFACTURE OF A MEDICAMENT FOR REDUCING...
https://pubmed.ncbi.nlm.nih.gov/28806222/
Transient Receptor Potential Vanilloid 1 Antagonists Prevent Anesthesia-induced Hypothermia and...
These studies demonstrate that transient receptor potential vanilloid 1 antagonists prevent anesthesia-induced hypothermia and decrease opioid dose...
transientreceptorpotential
https://pubchem.ncbi.nlm.nih.gov/bioassay/867
AID 867 - Counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput...
BioAssay record AID 867 submitted by The Scripps Research Institute Molecular Screening Center: Counterscreen for antagonists of galanin receptor 2 (GalR2): a...
https://bonndoc.ulb.uni-bonn.de/xmlui/handle/20.500.11811/10805
Irreversible Antagonists for the Adenosine A2B Receptor
for theirreversibleantagonistsadenosinereceptor